Gene information
Official symbol HTR2A
Official full name 5-hydroxytryptamine receptor 2A
Gene type protein-coding gene
Chromosome13q14.2
Alias symbol5-HT2A
Previous symbolHTR2
Gene family5-hydroxytryptamine receptors, G protein-coupled
Resources
Entrez Gene 3356
HGNC HGNC:5293
Ensembl ENSG00000102468
Vega OTTHUMG00000016881
UCSC uc010acr.5
GO terms: 153 records
GO Description Category LogP Number of genes Detail
GO:0001505 regulation of neurotransmitter levels GO Biological Processes -3.63969141 10 More
GO:0001618 virus receptor activity GO Molecular Functions -7.88412825 17 More
GO:0001659 temperature homeostasis GO Biological Processes -5.81640478 6 More
GO:0003012 muscle system process GO Biological Processes -27.3938503 63 More
GO:0003013 circulatory system process GO Biological Processes -65.2875605 130 More
GO:0003018 vascular process in circulatory system GO Biological Processes -47.1670528 52 More
GO:0005901 caveola GO Cellular Components -18.8033423 19 More
GO:0006109 regulation of carbohydrate metabolic process GO Biological Processes -13.1742479 35 More
GO:0006110 regulation of glycolytic process GO Biological Processes -6.41532756 12 More
GO:0006140 regulation of nucleotide metabolic process GO Biological Processes -7.41911571 18 More
GO:0006816 calcium ion transport GO Biological Processes -5.55009887 27 More
GO:0006874 cellular calcium ion homeostasis GO Biological Processes -8.17100062 15 More
GO:0006939 smooth muscle contraction GO Biological Processes -6.47455620 13 More
GO:0007187 G protein-coupled receptor signaling pathway, coupled to cyclic nucleotide second messenger GO Biological Processes -7.01019683 9 More
GO:0007200 phospholipase C-activating G protein-coupled receptor signaling pathway GO Biological Processes -11.6592522 24 More
GO:0007202 activation of phospholipase C activity GO Biological Processes -4.61361828 8 More
GO:0007268 chemical synaptic transmission GO Biological Processes -4.44678751 35 More
GO:0007610 behavior GO Biological Processes -18.1916656 76 More
GO:0007611 learning or memory GO Biological Processes -7.55755517 33 More
GO:0007613 memory GO Biological Processes -4.31484432 16 More
GO:0008015 blood circulation GO Biological Processes -65.7270163 119 More
GO:0009266 response to temperature stimulus GO Biological Processes -12.1149168 32 More
GO:0009410 response to xenobiotic stimulus GO Biological Processes -32.6021211 82 More
GO:0009581 detection of external stimulus GO Biological Processes -2.05740021 12 More
GO:0009582 detection of abiotic stimulus GO Biological Processes -2.39356289 13 More
GO:0009612 response to mechanical stimulus GO Biological Processes -18.7627330 44 More
GO:0009896 positive regulation of catabolic process GO Biological Processes -13.5088608 63 More
GO:0010517 regulation of phospholipase activity GO Biological Processes -7.06832255 9 More
GO:0010518 positive regulation of phospholipase activity GO Biological Processes -7.78358420 9 More
GO:0010863 positive regulation of phospholipase C activity GO Biological Processes -6.38368268 7 More
GO:0010959 regulation of metal ion transport GO Biological Processes -23.6318171 71 More
GO:0014065 phosphatidylinositol 3-kinase signaling GO Biological Processes -6.54430115 7 More
GO:0014829 vascular associated smooth muscle contraction GO Biological Processes -5.72938190 7 More
GO:0016032 viral process GO Biological Processes -8.84449931 34 More
GO:0016048 detection of temperature stimulus GO Biological Processes -2.54763391 5 More
GO:0017157 regulation of exocytosis GO Biological Processes -7.48561663 15 More
GO:0019058 viral life cycle GO Biological Processes -10.6409496 31 More
GO:0019216 regulation of lipid metabolic process GO Biological Processes -24.8423986 38 More
GO:0019229 regulation of vasoconstriction GO Biological Processes -25.9471687 22 More
GO:0019233 sensory perception of pain GO Biological Processes -10.7642352 20 More
GO:0019725 cellular homeostasis GO Biological Processes -21.1508273 85 More
GO:0030001 metal ion transport GO Biological Processes -7.54203733 26 More
GO:0030424 axon GO Cellular Components -6.14132550 54 More
GO:0030425 dendrite GO Cellular Components -4.55233052 48 More
GO:0030534 adult behavior GO Biological Processes -6.59104580 21 More
GO:0030594 neurotransmitter receptor activity GO Molecular Functions -2.67300750 6 More
GO:0031331 positive regulation of cellular catabolic process GO Biological Processes -13.5134767 30 More
GO:0033674 positive regulation of kinase activity GO Biological Processes -29.8538991 87 More
GO:0035150 regulation of tube size GO Biological Processes -44.5138102 41 More
GO:0035296 regulation of tube diameter GO Biological Processes -44.6572858 41 More
GO:0042310 vasoconstriction GO Biological Processes -9.70418585 13 More
GO:0043025 neuronal cell body GO Cellular Components -9.18558636 52 More
GO:0043235 receptor complex GO Cellular Components -19.4198369 40 More
GO:0043266 regulation of potassium ion transport GO Biological Processes -7.37974754 20 More
GO:0043267 negative regulation of potassium ion transport GO Biological Processes -7.26795046 12 More
GO:0043269 regulation of ion transport GO Biological Processes -36.9814668 116 More
GO:0043271 negative regulation of ion transport GO Biological Processes -19.3914052 40 More
GO:0043279 response to alkaloid GO Biological Processes -4.89883771 15 More
GO:0043405 regulation of MAP kinase activity GO Biological Processes -18.9267681 42 More
GO:0043408 regulation of MAPK cascade GO Biological Processes -57.2547066 142 More
GO:0043410 positive regulation of MAPK cascade GO Biological Processes -49.4744054 112 More
GO:0043467 regulation of generation of precursor metabolites and energy GO Biological Processes -10.8295915 27 More
GO:0043470 regulation of carbohydrate catabolic process GO Biological Processes -8.06132628 15 More
GO:0043549 regulation of kinase activity GO Biological Processes -36.8507249 123 More
GO:0044000 movement in host GO Biological Processes -9.40214314 25 More
GO:0044057 regulation of system process GO Biological Processes -61.6610386 136 More
GO:0044297 cell body GO Cellular Components -11.7206640 62 More
GO:0044409 entry into host GO Biological Processes -10.3666963 14 More
GO:0044853 plasma membrane raft GO Cellular Components -18.4542052 33 More
GO:0045121 membrane raft GO Cellular Components -30.0775030 71 More
GO:0045211 postsynaptic membrane GO Cellular Components -5.83105498 30 More
GO:0045598 regulation of fat cell differentiation GO Biological Processes -17.6607153 22 More
GO:0045600 positive regulation of fat cell differentiation GO Biological Processes -4.83398124 7 More
GO:0045821 positive regulation of glycolytic process GO Biological Processes -6.91942497 9 More
GO:0045834 positive regulation of lipid metabolic process GO Biological Processes -24.1838255 28 More
GO:0045859 regulation of protein kinase activity GO Biological Processes -34.3615088 109 More
GO:0045907 positive regulation of vasoconstriction GO Biological Processes -14.7401025 12 More
GO:0045913 positive regulation of carbohydrate metabolic process GO Biological Processes -10.1978214 20 More
GO:0045981 positive regulation of nucleotide metabolic process GO Biological Processes -9.35726225 15 More
GO:0046718 viral entry into host cell GO Biological Processes -10.4786216 14 More
GO:0046889 positive regulation of lipid biosynthetic process GO Biological Processes -14.1380112 16 More
GO:0046890 regulation of lipid biosynthetic process GO Biological Processes -16.6841590 23 More
GO:0048015 phosphatidylinositol-mediated signaling GO Biological Processes -5.56029805 8 More
GO:0048017 inositol lipid-mediated signaling GO Biological Processes -5.38623088 8 More
GO:0048871 multicellular organismal homeostasis GO Biological Processes -14.5562171 53 More
GO:0050433 regulation of catecholamine secretion GO Biological Processes -6.37680507 13 More
GO:0050730 regulation of peptidyl-tyrosine phosphorylation GO Biological Processes -27.1120967 60 More
GO:0050801 ion homeostasis GO Biological Processes -12.0812968 60 More
GO:0050804 modulation of chemical synaptic transmission GO Biological Processes -15.2260557 60 More
GO:0050805 negative regulation of synaptic transmission GO Biological Processes -5.05172294 12 More
GO:0050890 cognition GO Biological Processes -8.00500082 37 More
GO:0050951 sensory perception of temperature stimulus GO Biological Processes -3.21663541 6 More
GO:0050954 sensory perception of mechanical stimulus GO Biological Processes -4.15913068 20 More
GO:0050961 detection of temperature stimulus involved in sensory perception GO Biological Processes -3.03478521 5 More
GO:0050965 detection of temperature stimulus involved in sensory perception of pain GO Biological Processes -3.41433421 5 More
GO:0050982 detection of mechanical stimulus GO Biological Processes -3.60984508 9 More
GO:0051046 regulation of secretion GO Biological Processes -54.0079540 130 More
GO:0051051 negative regulation of transport GO Biological Processes -46.8709407 107 More
GO:0051209 release of sequestered calcium ion into cytosol GO Biological Processes -4.43542328 10 More
GO:0051282 regulation of sequestering of calcium ion GO Biological Processes -7.93009971 22 More
GO:0051283 negative regulation of sequestering of calcium ion GO Biological Processes -4.35719226 10 More
GO:0051345 positive regulation of hydrolase activity GO Biological Processes -19.7369783 79 More
GO:0051347 positive regulation of transferase activity GO Biological Processes -26.6059528 90 More
GO:0051588 regulation of neurotransmitter transport GO Biological Processes -2.92721908 6 More
GO:0051606 detection of stimulus GO Biological Processes -2.56190637 17 More
GO:0051701 biological process involved in interaction with host GO Biological Processes -10.6054189 28 More
GO:0051952 regulation of amine transport GO Biological Processes -10.5179624 22 More
GO:0051966 regulation of synaptic transmission, glutamatergic GO Biological Processes -5.51577792 8 More
GO:0055082 cellular chemical homeostasis GO Biological Processes -17.6289728 71 More
GO:0060191 regulation of lipase activity GO Biological Processes -10.2745708 13 More
GO:0060193 positive regulation of lipase activity GO Biological Processes -9.32996784 11 More
GO:0060627 regulation of vesicle-mediated transport GO Biological Processes -25.1756709 46 More
GO:0062012 regulation of small molecule metabolic process GO Biological Processes -26.8746473 69 More
GO:0062013 positive regulation of small molecule metabolic process GO Biological Processes -17.9792910 37 More
GO:0062149 detection of stimulus involved in sensory perception of pain GO Biological Processes -4.25041921 7 More
GO:0070372 regulation of ERK1 and ERK2 cascade GO Biological Processes -38.4320790 79 More
GO:0070374 positive regulation of ERK1 and ERK2 cascade GO Biological Processes -34.9831828 64 More
GO:0070588 calcium ion transmembrane transport GO Biological Processes -2.54626507 17 More
GO:0071407 cellular response to organic cyclic compound GO Biological Processes -19.6857751 39 More
GO:0071417 cellular response to organonitrogen compound GO Biological Processes -26.3253267 90 More
GO:0071867 response to monoamine GO Biological Processes -2.16454701 5 More
GO:0071868 cellular response to monoamine stimulus GO Biological Processes -2.21965331 5 More
GO:0071869 response to catecholamine GO Biological Processes -2.16454701 5 More
GO:0071870 cellular response to catecholamine stimulus GO Biological Processes -2.21965331 5 More
GO:0071900 regulation of protein serine/threonine kinase activity GO Biological Processes -19.5794055 63 More
GO:0090066 regulation of anatomical structure size GO Biological Processes -32.7608623 52 More
GO:0097447 dendritic tree GO Cellular Components -4.82959150 49 More
GO:0097553 calcium ion transmembrane import into cytosol GO Biological Processes -4.27502414 13 More
GO:0097746 blood vessel diameter maintenance GO Biological Processes -44.6572858 41 More
GO:0098655 cation transmembrane transport GO Biological Processes -3.98966777 20 More
GO:0098660 inorganic ion transmembrane transport GO Biological Processes -4.47276690 21 More
GO:0098662 inorganic cation transmembrane transport GO Biological Processes -4.65654157 20 More
GO:0098793 presynapse GO Cellular Components -4.56552653 42 More
GO:0098794 postsynapse GO Cellular Components -5.82876983 23 More
GO:0098857 membrane microdomain GO Cellular Components -30.8181788 72 More
GO:0098889 intrinsic component of presynaptic membrane GO Cellular Components -4.93822812 13 More
GO:0098916 anterograde trans-synaptic signaling GO Biological Processes -4.44678751 35 More
GO:0098978 glutamatergic synapse GO Cellular Components -4.83590061 31 More
GO:0099056 integral component of presynaptic membrane GO Cellular Components -4.69230219 12 More
GO:0099177 regulation of trans-synaptic signaling GO Biological Processes -15.1793607 60 More
GO:0099536 synaptic signaling GO Biological Processes -6.00976162 42 More
GO:0099537 trans-synaptic signaling GO Biological Processes -5.17038357 38 More
GO:0140272 exogenous protein binding GO Molecular Functions -8.63789613 18 More
GO:1900274 regulation of phospholipase C activity GO Biological Processes -6.23203613 7 More
GO:1900542 regulation of purine nucleotide metabolic process GO Biological Processes -7.57719972 18 More
GO:1900544 positive regulation of purine nucleotide metabolic process GO Biological Processes -9.35726225 15 More
GO:1901699 cellular response to nitrogen compound GO Biological Processes -26.9091664 96 More
GO:1903305 regulation of regulated secretory pathway GO Biological Processes -6.01402466 11 More
GO:1903522 regulation of blood circulation GO Biological Processes -44.9821911 79 More
GO:1903530 regulation of secretion by cell GO Biological Processes -45.6472055 114 More
GO:1903578 regulation of ATP metabolic process GO Biological Processes -8.20286273 19 More
GO:1903580 positive regulation of ATP metabolic process GO Biological Processes -9.55155535 14 More
GO:1903725 regulation of phospholipid metabolic process GO Biological Processes -3.02599739 4 More
KEGG pathways: 4 records
KEGG Description Category LogP Number of genes Detail
hsa04020 Calcium signaling pathway KEGG Pathway -10.4415222 36 More
hsa04080 Neuroactive ligand-receptor interaction KEGG Pathway -22.6219922 65 More
hsa04726 Serotonergic synapse KEGG Pathway -8.91693578 13 More
hsa04750 Inflammatory mediator regulation of TRP channels KEGG Pathway -4.64858532 8 More
Drug-Gene interaction
view
Related drugs: 101 records
Drug name Interaction type Source PMID View
abaperidone TTD view
amitriptyline antagonist TdgClinicalTrial 198009137855217 view
aniracetam TTD 11412837 view
aripiprazole partial agonistagonistantagonist TdgClinicalTrialChemblInteractionsTEND 17265076146429741724292526346901 view
aripiprazole lauroxil antagonist ChemblInteractions view
asenapine antagonist TdgClinicalTrial 183088142165534610592235 view
asenapine maleate antagonist ChemblInteractions view
bifeprunox TdgClinicalTrial view
blonanserin antagonist TTD 20030420 view
brexpiprazole antagonist TdgClinicalTrialChemblInteractions 24947465 view
bupropion PharmGKB 22947179 view
carphenazine maleate antagonist ChemblInteractions view
chlorpromazine binderantagonist ChemblInteractions 7908055859348410821438 view
chlorpromazine hydrochloride antagonist ChemblInteractions view
chlorprothixene antagonist TdgClinicalTrialChemblInteractionsTEND 28915503774629 view
citalopram PharmGKB 23158458195903973022179117671280 view
clozapine antagonist TdgClinicalTrialChemblInteractionsNCITENDPharmGKB 146878701453090315037867891610175209081297338524885933147514269926100 view
cyclobenzaprine antagonist TdgClinicalTrialTENDTTD 88842332197534912498911 view
cyclobenzaprine hydrochloride antagonist ChemblInteractions view
cyproheptadine antagonist TdgClinicalTrialTEND 12498911122338191641814914037901358088 view
doxepin antagonist TdgClinicalTrial 191799413091387855217 view
droperidol antagonist ChemblInteractions view
efavirenz PharmGKB 23859571 view
eplivanserin antagonist ChemblInteractions view
escitalopram inhibitor PharmGKB 1936539924424469 view
esmirtazapine inverse agonist TdgClinicalTrial 26047892 view
esmirtazapine maleate antagonist ChemblInteractions view
flibanserin antagonist TdgClinicalTrialTTD 264120541289070712177684 view
fluoxetine TdgClinicalTrial view
fluvoxamine PharmGKB 168740051620577719361869 view
haloperidol other/unknownantagonist ChemblInteractions 752090812629531 view
haloperidol decanoate antagonist ChemblInteractions view
haloperidol lactate antagonist ChemblInteractions view
iferanserin antagonist TdgClinicalTrialChemblInteractions view
iloperidone antagonist TdgClinicalTrialChemblInteractionsTTD 128614828997630 view
ketanserin inverse agonistantagonist NCI 976752417031071 view
lithium NCI 10758249 view
loxapine antagonist TdgClinicalTrialChemblInteractions 12664192 view
loxapine hydrochloride antagonist ChemblInteractions view
loxapine succinate antagonist ChemblInteractions view
lumateperone antagonist TdgClinicalTrialChemblInteractionsTTD 30596390 view
lurasidone antagonist TdgClinicalTrial 23545936 view
lurasidone hydrochloride antagonist ChemblInteractions view
mesoridazine antagonist TdgClinicalTrialTEND 115610661535795710991983 view
mesoridazine besylate antagonist ChemblInteractions view
methysergide antagonist TdgClinicalTrialTEND 1170465710080233117200801045528211061982 view
mianserin antagonist TdgClinicalTrialTEND 11004734 view
midomafetamine agonist TTD 28715817824160 view
minaprine antagonist TdgClinicalTrialTEND 3836113253009629752241361012 view
mirtazapine antagonist TdgClinicalTrialChemblInteractionsTEND 1706756015309042104467381160704711063897104467351044673410451911 view
molindone hydrochloride antagonist ChemblInteractions view
nefazodone antagonist TdgClinicalTrialTEND 7649970105776081287363214520130785521710435395909866310220119 view
nefazodone hydrochloride antagonist ChemblInteractions view
nelotanserin inverse agonist ChemblInteractionsTTD view
nemifitide TdgClinicalTrial view
ocaperidone TTD 10592235 view
olanzapine antagonist TdgClinicalTrialChemblInteractionsTENDPharmGKB 19193342145309031731670017848919158167871949444316905159117523521535897925032030248859331900094019636338324626991022711316038601 view
olanzapine pamoate antagonist ChemblInteractions view
ondansetron NCI 9767524 view
paliperidone antagonist TdgClinicalTrialChemblInteractionsTEND 11132243122110967520908752404375313537542676 view
paroxetine agonist PharmGKB 145144981825313423338224111366371140397758219561769739419361869 view
pimavanserin antagonistinverse agonist TdgClinicalTrialTTD 24016069 view
pimavanserin tartrate inverse agonist ChemblInteractions view
pimozide antagonist ChemblInteractions view
prochlorperazine TEND view
promazine antagonist TdgClinicalTrialTEND 1210677119110200109803251713928417016423 view
promazine hydrochloride antagonist ChemblInteractions view
propiomazine antagonist TdgClinicalTrialTEND 126786911911020017139284170164232250766414488364 view
pruvanserin antagonist ChemblInteractionsTTD view
quetiapine agonistantagonist TdgClinicalTrialTEND 1784891911132243175632571297338516038601 view
quetiapine fumarate antagonist ChemblInteractions view
renzapride TdgClinicalTrial view
risperdal TdgClinicalTrial view
risperidone antagonist TdgClinicalTrialChemblInteractionsTENDPharmGKB 159920902385957417316700111322431949444319997080259434581590715332462699 view
roluperidone hydrochloride TTD view
sarpogrelate inverse agonistantagonist TTD 1967203717031071 view
sb-773812 antagonist ChemblInteractions view
sertindole antagonist TdgClinicalTrialTEND 75302041692550811594443 view
sumatriptan PharmGKB 25096645 view
tedatioxetine antagonist ChemblInteractions view
temanogrel inverse agonist ChemblInteractionsTTD view
terguride agonist TdgClinicalTrial view
thiethylperazine TdgClinicalTrialTEND view
thioridazine antagonist TdgClinicalTrialChemblInteractionsTEND 86807349918563789877328662332423886 view
thioridazine hydrochloride antagonist ChemblInteractions view
thiothixene antagonist ChemblInteractions 859348410821438 view
thiothixene hydrochloride antagonist ChemblInteractions view
trazodone antagonist TdgClinicalTrialTEND 1059431630391201561092413656577855217117149001561457212782915 view
trazodone hydrochloride antagonist ChemblInteractions view
trelanserin antagonist TdgClinicalTrialChemblInteractions view
trifluoperazine hydrochloride antagonist ChemblInteractions view
trimipramine maleate antagonist ChemblInteractions view
tryptamine agonist TTD view
vabicaserin hydrochloride antagonist ChemblInteractions view
venlafaxine PharmGKB 22006095 view
volinanserin antagonist TdgClinicalTrialChemblInteractions view
zicronapine TTD view
ziprasidone antagonist TdgClinicalTrialTEND 17450180151216461253042311509214178489191244570514728084 view
ziprasidone hydrochloride antagonist ChemblInteractions view
ziprasidone mesylate antagonist ChemblInteractions view
zotepine antagonist TTD view
Related study: 1 record
Molecular factor Omics type Application Objective MI type Reference
NM_000621.5:c.102C>T genomics acute myocardial infarction[diagnosis] acute myocardial infarction Yamada S et al. Atherosclerosis. 2000
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